Copper catalysed amidation of aryl halides through chelation assistance.

نویسندگان

  • Subban Kathiravan
  • Shishir Ghosh
  • Graeme Hogarth
  • Ian A Nicholls
چکیده

A copper mediated C-N bond formation for the amidation of aryl halides using 8-aminoquinoline has been developed. This strategy provides efficient access to amides bearing two contiguous heterocyclic moieties and does not require the presence of additional ligands.

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عنوان ژورنال:
  • Chemical communications

دوره 51 23  شماره 

صفحات  -

تاریخ انتشار 2015